selected publications
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academic article
- A Selective Ligand for Estrogen Receptor Proteins Discriminates Rapid and Genomic Signaling.. Cell chemical biology. 26:1692-1702.e5. 2019
- G Protein-coupled Estrogen Receptor Protects from Atherosclerosis.. Scientific reports. 4:-. 2014
- GPER-targeted, 99mTc-labeled, nonsteroidal ligands demonstrate selective tumor imaging and in vivo estrogen binding.. Molecular cancer research : MCR. :-. 2014
- Synthesis and characterization of tricarbonyl-Re/Tc(I) chelate probes targeting the G protein-coupled estrogen receptor GPER/GPR30.. PloS one. 7:-. 2012
- Identification of a GPER/GPR30 antagonist with improved estrogen receptor counterselectivity.. The Journal of steroid biochemistry and molecular biology. 127:358-366. 2011
- Synthesis and characterization of iodinated tetrahydroquinolines targeting the G protein-coupled estrogen receptor GPR30.. Journal of medicinal chemistry. 53:1004-1014. 2010
- Highly efficient synthesis and characterization of the GPR30-selective agonist G-1 and related tetrahydroquinoline analogs.. Organic & biomolecular chemistry. 8:2252-2259. 2010
- Influence of charge on cell permeability and tumor imaging of GPR30-targeted 111in-labeled nonsteroidal imaging agents.. ACS chemical biology. 5:681-690. 2010
- In vivo effects of a GPR30 antagonist.. Nature chemical biology. 5:421-427. 2009
- Preclinical development of a neutral, estrogen receptor-targeted, tridentate 99mTc(I)-estradiol-pyridin-2-yl hydrazine derivative for imaging of breast and endometrial cancers.. Journal of nuclear medicine : official publication, Society of Nuclear Medicine. 49:978-986. 2008
- Synthetic estrogen derivatives demonstrate the functionality of intracellular GPR30.. ACS chemical biology. 2:536-544. 2007
- Linkage effects on binding affinity and activation of GPR30 and estrogen receptors ERalpha/beta with tridentate pyridin-2-yl hydrazine tricarbonyl-Re/(99m)Tc(I) chelates.. Journal of the American Chemical Society. 128:14476-14477. 2006
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document
- Erratum: G Protein-coupled Estrogen Receptor Protects from Atherosclerosis.. Scientific reports. -. 2015